SCHEMBL29967809

SCHEMBL29967809

CC(C)N1CC(CCNCc2cccc(Cl)c2)(c2ccccn2)CCC1=O

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 19/20 0.55
CYP2D6 P10635 4/20 0.53
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28272393 1.00 OPRM1 (0.55) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
Hydrochloric Acid SCHEMBL28868980 0.99 OPRM1 (0.54) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
Hydrochloric Acid SCHEMBL29967935 0.99 OPRM1 (0.54) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
SCHEMBL28270902 0.88 OPRM1 (0.57) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
SCHEMBL29968052 0.88 OPRM1 (0.57) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
Hydrochloric Acid SCHEMBL29968182 0.88 OPRM1 (0.56) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
Hydrochloric Acid SCHEMBL28272306 0.88 OPRM1 (0.56) OPRM1CYP2D6CYP3A4CYP2C19KCNH2
SCHEMBL28270851 0.77 OPRM1 (0.59) OPRM1CYP2D6CYP3A4KCNH2
Hydrochloric Acid SCHEMBL28271016 0.76 OPRM1 (0.58) OPRM1CYP2D6CYP3A4KCNH2
SCHEMBL28271045 0.76 GRIN1 (0.34) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109206417-B Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2023-01-03 CN disclosed
CN-115124520-A Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2022-09-30 CN disclosed