SCHEMBL29968423

SCHEMBL29968423

Nc1n[nH]c2cccc(-c3ccc(C(F)(F)F)cc3)c12

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.71
ABL1 P00519 7/20 0.71
LCK P06239 4/20 0.71
CSF1R P07333 4/20 0.71
FGFR1 P11362 3/20 0.71
PRKACA P17612 3/20 0.71
ROCK1 Q13464 3/20 0.71
FLT1 P17948 3/20 0.71
NTRK1 P04629 2/20 0.71
MET P08581 2/20 0.71
GSK3A P49840 2/20 0.71
GSK3B P49841 2/20 0.71
RPS6KA3 P51812 2/20 0.71
CDK5 Q00535 2/20 0.71
DYRK1A Q13627 2/20 0.71
DAPK3 O43293 1/20 0.71
PRKD3 O94806 1/20 0.71
MAP4K4 O95819 1/20 0.71
PAK4 O96013 1/20 0.71
RET P07949 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16681039 1.00 KDR (0.71) KDRABL1LCKCSF1RFGFR1
SCHEMBL6013181 0.87 KDR (0.90) KDRABL1LCKCSF1RFGFR1
SCHEMBL29968383 0.85 KDR (0.70) KDRABL1LCKCSF1RFGFR1
SCHEMBL28957310 0.85 KDR (0.70) KDRABL1LCKCSF1RFGFR1
SCHEMBL31060697 0.83 KDR (1.00) KDRABL1LCKCSF1RFGFR1
SCHEMBL421242 0.83 KDR (1.00) KDRABL1LCKCSF1RFGFR1
SCHEMBL28871225 0.82 KDR (0.74) KDRABL1LCKCSF1RFGFR1
SCHEMBL29967675 0.82 KDR (0.74) KDRABL1LCKCSF1RFGFR1
SCHEMBL1383263 0.82 KDR (0.69) KDRABL1LCKCSF1RFGFR1
SCHEMBL10213956 0.81 KDR (0.73) KDRABL1LCKCSF1RFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed