SCHEMBL29968893

SCHEMBL29968893

Cn1nc(N)c2c(-c3ccc(C(C)(C)C)cc3)cccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.52
FLT3 P36888 5/20 0.52
CSF1R P07333 4/20 0.47
KIT P10721 4/20 0.47
FLT1 P17948 4/20 0.47
FLT4 P35916 4/20 0.47
LCK P06239 3/20 0.47
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
DGAT1 O75907 2/20 0.42
S1PR1 P21453 1/20 0.42
LYN P07948 3/20 0.41
BLK P51451 3/20 0.41
DYRK3 O43781 2/20 0.41
ROCK2 O75116 2/20 0.41
MAP4K4 O95819 2/20 0.41
RET P07949 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28871229 1.00 KDR (0.52) KDRFLT3CSF1RKITFLT1
SCHEMBL422378 0.85 KDR (0.56) KDRFLT3CSF1RKITFLT1
SCHEMBL29968188 0.78 KDR (0.46) KDRFLT3CSF1RKITFLT1
SCHEMBL28871314 0.78 KDR (0.46) KDRFLT3CSF1RKITFLT1
SCHEMBL28871230 0.76 MAP2K4 (0.44) KDRFLT3CSF1RKITFLT1
SCHEMBL29967811 0.76 MAP2K4 (0.44) KDRFLT3CSF1RKITFLT1
SCHEMBL1384538 0.76 KDR (0.71) KDRFLT3CSF1RKITFLT1
SCHEMBL28871271 0.74 CYP2C9 (0.51) KDRFLT3NPC1TP53RAB9A
SCHEMBL422432 0.73 KDR (0.82) KDRFLT3CSF1RKITFLT1
SCHEMBL424772 0.72 KDR (0.84) KDRFLT3CSF1RKITFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed