SCHEMBL29970923

SCHEMBL29970923

COC(=O)CCc1cccc(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.53
SIRT2 Q8IXJ6 1/20 0.51
FFAR1 O14842 2/20 0.50
FFAR4 Q5NUL3 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
ESR1 P03372 1/20 0.49
NR3C1 P04150 1/20 0.49
PGR P06401 1/20 0.49
NR3C2 P08235 1/20 0.49
AR P10275 1/20 0.49
THRA P10827 1/20 0.49
THRB P10828 1/20 0.49
PTPN1 P18031 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
IDO1 P14902 1/20 0.46
PTGES O14684 1/20 0.46
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6378 1.00 TAAR1 (0.53) TAAR1SIRT2FFAR1FFAR4L3MBTL1
SCHEMBL7109146 0.90 TAAR1 (0.50) TAAR1FFAR1FFAR4PTGES
Phenyl Propionic Acid SCHEMBL28549085 0.90 FFAR1 (0.59) SIRT2FFAR1FFAR4L3MBTL1ESR1
SCHEMBL1743642 0.85 FFAR1 (0.74) FFAR1FFAR4ESR1NR3C1PGR
SCHEMBL1511063 0.84 CYP4F2 (0.55) TAAR1FFAR1FFAR4L3MBTL1ESR1
SCHEMBL15504971 0.83 SIRT2 (0.51) SIRT2PTPN1
SCHEMBL26714888 0.83 FFAR1 (0.50) TAAR1FFAR1FFAR4L3MBTL1ESR1
SCHEMBL29700723 0.83 SLC7A5 (0.55) TAAR1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL136054 0.83 SLC7A5 (0.55) TAAR1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL902744 0.83 L3MBTL1 (0.47) TAAR1FFAR1FFAR4L3MBTL1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115279747-B FYN and VEGFR2 kinase inhibitors 罗达制药生物技术有限责任公司 2024-11-05 CN disclosed
CN-115279747-A Novel fYN and VEGFR2 kinase inhibitors 罗达制药生物技术有限责任公司 2022-11-01 CN disclosed