SCHEMBL29972701

SCHEMBL29972701

Cc1cn(-c2ccc(Br)cn2)nn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
LRRK2 Q5S007 1/20 0.38
ALDH1A1 P00352 2/20 0.38
P2RX7 Q99572 1/20 0.38
GRIN1 Q05586 3/20 0.36
GRIN2B Q13224 3/20 0.36
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
KCNJ1 P48048 1/20 0.35
EGLN2 Q96KS0 1/20 0.35
KDM4E B2RXH2 2/20 0.34
NOTUM Q6P988 1/20 0.34
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13430089 1.00 BRD4 (0.39) BRD4LRRK2ALDH1A1P2RX7GRIN1
SCHEMBL23999584 0.82 LRRK2 (0.47) BRD4LRRK2GRIN1GRIN2BGRIN2D
SCHEMBL25045462 0.79 NOTUM (0.40) BRD4LRRK2ALDH1A1GRIN1GRIN2B
SCHEMBL20639984 0.77 P2RX7 (0.47) ALDH1A1P2RX7GRIN1GRIN2BGRIN2D
SCHEMBL20168136 0.77 EGLN2 (0.46) BRD4LRRK2GRIN1GRIN2BKCNJ1
SCHEMBL30751809 0.77 EGLN2 (0.46) BRD4LRRK2GRIN1GRIN2BKCNJ1
SCHEMBL4555166 0.76 CYP1A2 (0.47) LRRK2ALDH1A1P2RX7GRIN1GRIN2B
SCHEMBL25043785 0.76 GRIN1 (0.40) BRD4LRRK2GRIN1GRIN2BKCNJ1
SCHEMBL24135300 0.76 BRD4 (0.40) BRD4LRRK2ALDH1A1GRIN1GRIN2B
SCHEMBL30445199 0.76 KCNJ1 (0.55) BRD4LRRK2ALDH1A1P2RX7GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114845778-A Dihydrocyclopentaisoquinoline sulfonamide derivative compound UCB生物制药有限责任公司 2022-08-02 CN disclosed