SCHEMBL29976559

SCHEMBL29976559

CC(=O)c1cnc(Nc2ccc3c(=O)cc(C(F)(F)F)n(C)c3c2)s1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.50
RAB9A P51151 4/20 0.50
NPC1 O15118 2/20 0.49
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
DHODH Q02127 2/20 0.37
KMT2A Q03164 1/20 0.37
MAPK13 O15264 2/20 0.35
MAPK12 P53778 2/20 0.35
MAPK11 Q15759 2/20 0.35
MAPK14 Q16539 2/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CDK5 Q00535 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29976542 0.92 SMN1; SMN2 (0.41) SMN1; SMN2RAB9ANPC1KDM4EALDH1A1
SCHEMBL29977188 0.92 SMN1; SMN2 (0.40) SMN1; SMN2RAB9ANPC1KDM4EALDH1A1
SCHEMBL29977036 0.86 SMN1; SMN2 (0.36) SMN1; SMN2RAB9ANPC1KDM4EALDH1A1
SCHEMBL29977354 0.85 CSNK2A2 (0.35) SMN1; SMN2RAB9ANPC1KMT2A
SCHEMBL29976800 0.85 SMN1; SMN2 (0.36) SMN1; SMN2RAB9ANPC1KDM4EALDH1A1
SCHEMBL29977250 0.84 IRAK4 (0.35) SMN1; SMN2RAB9ANPC1
SCHEMBL29976735 0.83 SCD (0.37) SMN1; SMN2KDM4EALDH1A1HPGDKMT2A
SCHEMBL29976557 0.83 PSEN1 (0.33) SMN1; SMN2RAB9ANPC1CCNE1CDK2
SCHEMBL29977028 0.82 KDR (0.38)
SCHEMBL29977049 0.81 GAA (0.32) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403558-A Aromatic heterocyclic compound with antitumor activity and preparation method and application thereof 河南真实生物科技有限公司 2022-11-29 CN disclosed