SCHEMBL29976557

SCHEMBL29976557

CC(O)c1cnc(Nc2ccc3c(=O)cc(C(F)(F)F)n(C)c3c2)s1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
PKM P14618 1/20 0.32
PKLR P30613 1/20 0.32
ALPL P05186 1/20 0.32
ALPI P09923 1/20 0.32
CDK2 P24941 2/20 0.31
CCNE1 P24864 1/20 0.31
CDK5 Q00535 1/20 0.31
RAB9A P51151 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29977354 0.84 CSNK2A2 (0.35) PKMPKLRRAB9ASMN1; SMN2NPC1
SCHEMBL29977188 0.83 SMN1; SMN2 (0.40) RAB9ASMN1; SMN2NPC1
SCHEMBL29976559 0.83 SMN1; SMN2 (0.50) CDK2CCNE1CDK5RAB9ASMN1; SMN2
SCHEMBL29976542 0.83 SMN1; SMN2 (0.41) RAB9ASMN1; SMN2NPC1
SCHEMBL29977250 0.83 IRAK4 (0.35) PKMPKLRALPLALPIRAB9A
SCHEMBL29977028 0.81 KDR (0.38)
SCHEMBL29976735 0.80 SCD (0.37) ALPLALPISMN1; SMN2
SCHEMBL29976548 0.78 PLA2G7 (0.41) PKMRAB9ASMN1; SMN2NPC1
SCHEMBL29977049 0.78 GAA (0.32) SMN1; SMN2
SCHEMBL29976739 0.78 ALPL (0.35) ALPLALPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403558-A Aromatic heterocyclic compound with antitumor activity and preparation method and application thereof 河南真实生物科技有限公司 2022-11-29 CN disclosed