SCHEMBL29977346

SCHEMBL29977346

Cn1c(C(N)=O)cc(=O)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.53
EGFR P00533 2/20 0.50
SRC P12931 1/20 0.50
ERCC1 P07992 1/20 0.47
FEN1 P39748 1/20 0.47
ERCC4 Q92889 1/20 0.47
KDM4E B2RXH2 6/20 0.45
ALDH1A1 P00352 5/20 0.45
HSD17B10 Q99714 5/20 0.45
CYP2C19 P33261 2/20 0.45
LMNA P02545 2/20 0.45
NQO2 P16083 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
HIF1A Q16665 1/20 0.45
SLC9A1 P19634 2/20 0.44
GPR3 P46089 1/20 0.44
MCL1 Q07820 1/20 0.44
GLA P06280 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27730322 0.85 MCL1 (0.62) HPGDEGFRSRCERCC1FEN1
SCHEMBL29618419 0.83 HPGD (0.53) HPGDERCC1FEN1ERCC4KDM4E
SCHEMBL19249104 0.81 KDM4E (0.53) HPGDEGFRSRCERCC1FEN1
SCHEMBL28254849 0.80 HPGD (0.38) HPGDEGFRSRCERCC1FEN1
SCHEMBL31257225 0.80 POLB (0.47) HPGDEGFRSRCALDH1A1CYP2C19
SCHEMBL8201715 0.79 SLC9A1 (0.50) HPGDEGFRSRCKDM4EALDH1A1
SCHEMBL2323444 0.77 MCL1 (0.71) SLC9A1MCL1NPC1
SCHEMBL11186759 0.77 KDM4E (0.58) HPGDKDM4EALDH1A1HSD17B10LMNA
SCHEMBL5005344 0.77 SLC9A1 (0.51) EGFRSRCKDM4EALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL28264080 0.76 MCL1 (0.69) SLC9A1MCL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403558-A Aromatic heterocyclic compound with antitumor activity and preparation method and application thereof 河南真实生物科技有限公司 2022-11-29 CN disclosed