SCHEMBL29978028

SCHEMBL29978028

N#Cc1ccc(C(=O)N2CCc3sc(-c4noc(C(F)(F)F)n4)cc3C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 10/20 0.47
HDAC6 Q9UBN7 5/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC2 Q92769 1/20 0.47
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
GRM5 P41594 1/20 0.38
STAT3 P40763 1/20 0.37
PRLHR P49683 3/20 0.37
HDAC1 Q13547 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
SLC9A1 P19634 1/20 0.37
CYP2C19 P33261 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978914 0.89 HDAC4 (0.50) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29978582 0.89 HDAC4 (0.50) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29977967 0.89 HDAC4 (0.50) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29978301 0.88 HDAC4 (0.52) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29978909 0.88 HDAC4 (0.48) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29978387 0.88 HDAC4 (0.50) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29978396 0.86 HDAC4 (0.48) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29978536 0.86 HDAC4 (0.49) HDAC4HDAC6HDAC8HDAC2PRMT5
SCHEMBL29977801 0.85 HDAC4 (0.39) HDAC4HDAC6HDAC8HDAC2GRM5
SCHEMBL29978118 0.84 HDAC4 (0.45) HDAC4HDAC6HDAC8HDAC2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed