SCHEMBL29978653

SCHEMBL29978653

OCc1ccnc(OCC(F)F)n1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RXRA P19793 18/20 0.46
GRIN1 Q05586 18/20 0.46
GRIN2B Q13224 18/20 0.46
CCR1 P32246 1/20 0.34
SORD Q00796 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16815492 0.77 RXRA (0.42) RXRAGRIN1GRIN2BCCR1SORD
SCHEMBL16815816 0.76 RXRA (0.43) RXRAGRIN1GRIN2BCCR1
SCHEMBL21910852 0.75 RXRA (0.42) RXRAGRIN1GRIN2B
SCHEMBL16815694 0.74 CCR1 (0.39) RXRAGRIN1GRIN2BCCR1
SCHEMBL16815642 0.74 MAPK8 (0.44) RXRAGRIN1GRIN2BCCR1
SCHEMBL16815405 0.74 RXRA (0.41) RXRAGRIN1GRIN2BCCR1SORD
SCHEMBL20745081 0.73 RXRA (0.37) RXRAGRIN1GRIN2BCCR1
SCHEMBL16815518 0.73 RXRA (0.41) RXRAGRIN1GRIN2BCCR1
SCHEMBL16815225 0.72 RXRA (0.38) RXRAGRIN1GRIN2BCCR1
SCHEMBL16815693 0.71 RXRA (0.45) RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022216945-A1 MACROCYCLIC MCL1 INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-10-13 WO disclosed