SCHEMBL29979185

SCHEMBL29979185

Cc1c(Br)cc(Cl)c(O)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 5/20 0.37
HIF1A Q16665 3/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ALOX15 P16050 2/20 0.37
ALOX12 P18054 2/20 0.37
CYP1A2 P05177 1/20 0.37
TSHR P16473 5/20 0.36
CYP3A4 P08684 3/20 0.36
TTR P02766 2/20 0.36
ALDH1A1 P00352 2/20 0.36
RECQL P46063 2/20 0.36
HPGD P15428 3/20 0.33
THRB P10828 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SIRT1 Q96EB6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL524725 0.80 CA1 (0.42) HSD17B10HIF1ASMN1; SMN2ALOX15ALOX12
SCHEMBL3029667 0.78 HSD17B10 (0.46) HSD17B10HIF1ACYP2C9CYP2C19SMN1; SMN2
SCHEMBL23304085 0.78 CYP3A4 (0.33) HSD17B10HIF1AALOX15ALOX12TSHR
SCHEMBL9051494 0.76 TSHR (0.40) HSD17B10HIF1ACYP2C9CYP2C19SMN1; SMN2
SCHEMBL24161857 0.76 KDM1A (0.32) KDM1AKDM1B
SCHEMBL24727674 0.76 HSD17B10 (0.40) HSD17B10HIF1ACYP2C9CYP2C19SMN1; SMN2
SCHEMBL3822643 0.75 CA1 (0.37) CYP3A4ALDH1A1MAPTTDP1KDM1A
SCHEMBL25924982 0.72 SIRT1 (0.41) HSD17B10HIF1ACYP2C9CYP2C19SMN1; SMN2
SCHEMBL31026375 0.71 TSHR (0.31) TSHRNQO2KDM1AKDM1B
SCHEMBL21186739 0.71 HSD17B10 (0.42) HSD17B10HIF1ACYP2C9CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022216945-A1 MACROCYCLIC MCL1 INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-10-13 WO disclosed