SCHEMBL29987229

SCHEMBL29987229

NC(=O)c1ccc(N2CCNCC2)nc1Oc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 14/20 0.70
CYP2C8 P10632 1/20 0.52
KCNH2 Q12809 1/20 0.52
LTA4H P09960 1/20 0.49
KDM4E B2RXH2 2/20 0.48
CYP3A4 P08684 2/20 0.48
HSD17B10 Q99714 2/20 0.48
HTR3E A5X5Y0 1/20 0.45
USP2 O75604 1/20 0.45
HTR3B O95264 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
ADRB1 P08588 1/20 0.45
HTR1A P08908 1/20 0.45
HTR2C P28335 1/20 0.45
MAPK1 P28482 1/20 0.45
SLC6A4 P31645 1/20 0.45
HTR7 P34969 1/20 0.45
HTT P42858 1/20 0.45
HTR3A P46098 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28881569 1.00 BTK (0.70) BTKCYP2C8KCNH2LTA4HKDM4E
Hydrochloric Acid SCHEMBL16671009 0.99 BTK (0.69) BTKCYP2C8KCNH2LTA4HKDM4E
SCHEMBL20998572 0.88 BTK (0.72) BTKCYP2C8KCNH2
SCHEMBL16597779 0.86 BTK (0.71) BTKLTA4HSCN9A
SCHEMBL16670516 0.82 BTK (1.00) BTKCYP2C8KCNH2
SCHEMBL16676723 0.82 BTK (0.48) BTKLTA4HCYP3A4HSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL16670652 0.81 BTK (0.48) BTKLTA4HUSP2CYP1A2MAPK8
SCHEMBL28881829 0.81 BTK (0.68) BTKCYP2C8KCNH2
SCHEMBL16676769 0.81 BTK (0.68) BTKCYP2C8KCNH2
SCHEMBL29987334 0.81 BTK (0.68) BTKCYP2C8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304606-B Degradation agent for simultaneously targeting BTK and GSPT proteins 清华大学 2024-04-19 CN disclosed
CN-115304606-A Degradation agent for simultaneously targeting BTK and GSPT1 proteins 清华大学 2022-11-08 CN disclosed