SCHEMBL29987481

SCHEMBL29987481

O=C(NC1CCNCC1)c1cccc2c[nH]cc12

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.53
CDK9 P50750 1/20 0.53
CDK5 Q00535 1/20 0.53
CDK5R1 Q15078 1/20 0.53
PARP1 P09874 2/20 0.49
HTR4 Q13639 2/20 0.47
DRD4 P21917 6/20 0.46
KMT2A Q03164 1/20 0.46
CHEK1 O14757 1/20 0.46
CDK2 P24941 1/20 0.45
CCNA1 P78396 1/20 0.45
P2RX7 Q99572 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
PBK Q96KB5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31074994 0.86 KMT2A (0.61) DRD4KMT2A
SCHEMBL62620 0.86 KMT2A (0.61) DRD4KMT2A
Hydrochloric Acid SCHEMBL3160630 0.84 KMT2A (0.60) DRD4KMT2A
SCHEMBL27511688 0.77 KMT2A (0.49) CCNT1CDK9CDK5CDK5R1PARP1
SCHEMBL5038597 0.77 KEAP1 (0.51) CCNT1CDK9CDK5CDK5R1PARP1
SCHEMBL8124625 0.76 PARP1 (0.47) CCNT1CDK9CDK5CDK5R1PARP1
SCHEMBL31465178 0.75 NPC1 (0.71) CCNT1CDK9CDK5CDK5R1PARP1
Hydrochloric Acid SCHEMBL23360011 0.75 PARP1 (0.52) CCNT1CDK9CDK5CDK5R1PARP1
SCHEMBL28917070 0.75 CDK2 (0.56) CCNT1CDK9CDK5CDK5R1PARP1
SCHEMBL30088642 0.75 TNKS (0.55) CCNT1CDK9CDK5CDK5R1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304606-B Degradation agent for simultaneously targeting BTK and GSPT proteins 清华大学 2024-04-19 CN disclosed
CN-115304606-A Degradation agent for simultaneously targeting BTK and GSPT1 proteins 清华大学 2022-11-08 CN disclosed