SCHEMBL299929

SCHEMBL299929

c1ccc(C2CCC3CCCCN3C2)cc1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.68
CYP2C19 P33261 1/20 0.68
SLC18A3 Q16572 1/20 0.62
HPGD P15428 1/20 0.53
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HRH3 Q9Y5N1 1/20 0.51
GRIN2B Q13224 2/20 0.46
MBTD1 Q05BQ5 1/20 0.46
L3MBTL3 Q96JM7 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GRIN1 Q05586 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27894548 0.95 CYP2D6 (0.65) CYP2D6CYP2C19SLC18A3HPGDKMT2A
SCHEMBL13660519 0.86 SLC18A3 (0.57) CYP2D6CYP2C19SLC18A3SMN1; SMN2
SCHEMBL28702035 0.84 CYP2D6 (0.93) CYP2D6CYP2C19SLC18A3HPGDKMT2A
SCHEMBL24163290 0.84 SLC18A3 (0.79) CYP2D6CYP2C19SLC18A3HPGDKMT2A
SCHEMBL14720645 0.82 SLC18A3 (0.83) CYP2D6CYP2C19SLC18A3HPGDKMT2A
SCHEMBL22794986 0.82 SLC18A3 (0.53) CYP2D6CYP2C19SLC18A3HRH3
SCHEMBL22794978 0.82 SLC18A3 (0.53) CYP2D6CYP2C19SLC18A3HRH3
SCHEMBL22795507 0.82 SLC18A3 (0.53) CYP2D6CYP2C19SLC18A3HRH3
SCHEMBL24877147 0.82 SLC18A3 (0.70) CYP2D6CYP2C19SLC18A3HPGDKMT2A
SCHEMBL15184744 0.82 CYP2D6 (0.83) CYP2D6CYP2C19SLC18A3HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888604-B1 PROCESS FOR PREPARING (ALPHA S, BETA R)-6-BROMO-ALPHA-[2-(DIMETHYLAMINO)ETHYL]-2-METHOXY-ALPHA-1-NAPHTHALENYL-BETA-PHENYL-3-QUINOLINEETHANOL JANSSEN PHARMACEUTICA NV (BE) 2012-03-14 EP disclosed
EP-0012170-A1 7-Phenyl-quinolizidine derivatives (I), their preparation, pharmaceutical compositions containing them and (I) for use in treating diseases F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1980-06-25 EP disclosed