SCHEMBL29995286

SCHEMBL29995286

FC(F)(F)Oc1ccc(Oc2ccnc3ccccc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.52
BRAF P15056 1/20 0.52
MAPK14 Q16539 1/20 0.52
TNNI3K Q59H18 1/20 0.52
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
ERBB2 P04626 1/20 0.43
RAF1 P04049 1/20 0.42
LCK P06239 1/20 0.42
RET P07949 1/20 0.42
CYP3A4 P08684 1/20 0.42
KIT P10721 1/20 0.42
MAP3K20 Q9NYL2 1/20 0.42
RIPK3 Q9Y572 1/20 0.42
FGFR2 P21802 3/20 0.41
ACP1 P24666 1/20 0.41
AXL P30530 2/20 0.40
KCNH2 Q12809 1/20 0.40
SCN5A Q14524 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27303568 0.83 KDR (0.49) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL1897179 0.82 ERBB2 (0.55) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL7468525 0.80 MAPT (0.49) KDRFGFR2PDGFRBPDGFRA
SCHEMBL12386844 0.80 KDR (0.48) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL1546587 0.80 KDM1A (0.54) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL29812245 0.80 KDM1A (0.54) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL29802752 0.80 KDR (0.55) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL29269610 0.79 ACP1 (0.47) KDRMAPK14RAF1LCKRET
SCHEMBL9431770 0.78 NCF1 (0.54) KDRBRAFMAPK14TNNI3KERBB2
SCHEMBL7462207 0.77 NR4A2 (0.44) KDRBRAFMAPK14TNNI3KSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115210225-A Substituted aminoquinolones as immuno-activated DGKALPHA inhibitors 拜耳公司 2022-10-18 CN disclosed