SCHEMBL299959

SCHEMBL299959

CS(=O)(=O)c1ccc2c(c1)CCN2c1cc(OC2CCN(C(=O)O)CC2)ncn1

nearest known ligand 0.80

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 20/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL515140 0.92 GPR119 (0.76) GPR119
SCHEMBL515139 0.92 GPR119 (0.79) GPR119
SCHEMBL2717368 0.92 GPR119 (0.72) GPR119
SCHEMBL10255383 0.91 GPR119 (0.84) GPR119
SCHEMBL17091636 0.91 GPR119 (0.67) GPR119
SCHEMBL3238465 0.91 GPR119 (0.77) GPR119
SCHEMBL3237856 0.91 GPR119 (0.74) GPR119
SCHEMBL3511634 0.90 GPR119 (0.81) GPR119
SCHEMBL3242159 0.90 GPR119 (0.79) GPR119
SCHEMBL3238021 0.90 GPR119 (0.75) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2210886-B1 PYRIMIDYL INDOLINE COMPOUND DAIICHI SANKYO CO LTD (JP) 2015-09-23 EP claimed
EP-2445901-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO Boehringer Ingelheim International GmbH (DE) 2012-05-02 EP disclosed
EP-2427450-A1 GPR 119 MODULATORS Pfizer Inc. (US) 2012-03-14 EP disclosed
WO-2010149685-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-29 WO disclosed
WO-2010128425-A1 GPR 119 MODULATORS PFIZER INC. (US) 2010-11-11 WO disclosed