SCHEMBL29997804

SCHEMBL29997804

COc1ccc(COc2cc(N3C[C@@H](C)O[C@H](C)C3)cc(Cl)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 5/20 0.45
PDE2A O00408 1/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 4/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
NPC1 O15118 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RAB9A P51151 2/20 0.37
FGFR1 P11362 1/20 0.37
FGFR2 P21802 1/20 0.37
FGFR3 P22607 1/20 0.37
KDR P35968 1/20 0.37
HPGD P15428 1/20 0.37
MDM2 Q00987 1/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23459340 1.00 PDE1B (0.45) PDE1BPDE2ATSHRNPSR1KMT2A
SCHEMBL25698372 0.88 PDE2A (0.41) PDE1BPDE2ANPC1RAB9ALRRK2
SCHEMBL29998665 0.88 PDE2A (0.41) PDE1BPDE2ANPC1RAB9ALRRK2
SCHEMBL23459396 0.88 PDE2A (0.41) PDE1BPDE2ANPC1RAB9ALRRK2
SCHEMBL23477942 0.88 DRD4 (0.40) PDE1BPDE2AL3MBTL1HPGDMAPT
SCHEMBL29997749 0.82 MAPT (0.51) PDE2ANPSR1ALDH1A1L3MBTL1RAB9A
SCHEMBL17819740 0.82 MAPT (0.51) PDE2ANPSR1ALDH1A1L3MBTL1RAB9A
SCHEMBL23477951 0.80 PDE2A (0.36) PDE1BPDE2ANPC1RAB9A
SCHEMBL23459240 0.78 DRD4 (0.37) PDE2AL3MBTL1MAPTGRM2
SCHEMBL29997788 0.78 DRD4 (0.37) PDE2AL3MBTL1MAPTGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4069366-A1 ATM KINASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI Foundation, Inc. (US) 2022-10-12 EP disclosed