SCHEMBL30000717

SCHEMBL30000717

COC(=O)c1cc(NC2CCN(C(C)=O)CC2)nc(O)n1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.45
MAPT P10636 1/20 0.42
QDPR P09417 1/20 0.40
PRMT5 O14744 3/20 0.40
WDR77 Q9BQA1 1/20 0.40
NOS2 P35228 7/20 0.39
NOS1 P29475 6/20 0.39
NOS3 P29474 3/20 0.39
HPGDS O60760 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
CDK2 P24941 1/20 0.39
REV1 Q9UBZ9 2/20 0.39
DYRK1A Q13627 1/20 0.38
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25389761 1.00 NSD2 (0.45) NSD2MAPTQDPRPRMT5WDR77
SCHEMBL25388838 0.88 NSD2 (0.43) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL30000062 0.88 NSD2 (0.43) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL29501351 0.87 NSD2 (0.42) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL22549439 0.87 NSD2 (0.42) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL27172393 0.85 NSD2 (0.45) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL29999584 0.85 NSD2 (0.45) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL27172459 0.85 MAPT (0.45) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL30000118 0.85 MAPT (0.45) NSD2MAPTPRMT5WDR77NOS2
SCHEMBL23304428 0.84 GBA1 (0.46) NSD2MAPTPRMT5WDR77NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116113626-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2023-05-12 CN disclosed
WO-2022237858-A1 COMPOUND HAVING ANTI-TUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-11-17 WO disclosed
CN-115340528-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2022-11-15 CN disclosed