SCHEMBL29501351

SCHEMBL29501351

COC(=O)c1cc(NC2CCN(C(C)=O)CC2)nc(Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.42
NOS2 P35228 7/20 0.42
NOS1 P29475 6/20 0.42
NOS3 P29474 4/20 0.41
MAPT P10636 1/20 0.41
PRMT5 O14744 3/20 0.39
WDR77 Q9BQA1 1/20 0.39
HPGDS O60760 1/20 0.39
PDCD1LG2 Q9BQ51 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
CDK1 P06493 1/20 0.38
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CDK2 P24941 1/20 0.38
REV1 Q9UBZ9 2/20 0.38
DYRK1A Q13627 1/20 0.38
SYK P43405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22549439 1.00 NSD2 (0.42) NSD2NOS2NOS1NOS3MAPT
SCHEMBL22418701 0.88 NOS1 (0.41) NSD2NOS2NOS1NOS3MAPT
SCHEMBL23304536 0.88 FLT3 (0.41) PRMT5WDR77SYK
SCHEMBL30000062 0.87 NSD2 (0.43) NSD2NOS2NOS1NOS3MAPT
SCHEMBL25389761 0.87 NSD2 (0.45) NSD2NOS2NOS1NOS3MAPT
SCHEMBL25388838 0.87 NSD2 (0.43) NSD2NOS2NOS1NOS3MAPT
SCHEMBL30000717 0.87 NSD2 (0.45) NSD2NOS2NOS1NOS3MAPT
Hydrochloric Acid SCHEMBL25387169 0.87 NOS1 (0.40) NSD2NOS2NOS1NOS3MAPT
Hydrochloric Acid SCHEMBL29501501 0.87 NOS1 (0.40) NSD2NOS2NOS1NOS3MAPT
SCHEMBL1748149 0.85 ALDH1A1 (0.51) NSD2NOS2NOS1MAPTDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110621675-B Tricyclic compounds useful for the treatment of proliferative diseases 阿古诺治疗有限公司 2023-09-19 CN disclosed
CN-116113626-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2023-05-12 CN disclosed
CN-115340528-A Compound with anti-tumor activity and application thereof 上海翊石医药科技有限公司 2022-11-15 CN disclosed
WO-2022048631-A1 COMPOUND HAVING ANTITUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-03-10 WO disclosed