SCHEMBL30000766

SCHEMBL30000766

Cc1cc(N)nc(C)c1CN

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 6/20 0.41
NOS2 P35228 6/20 0.41
NOS1 P29475 5/20 0.41
BACE1 P56817 1/20 0.38
KLKB1 P03952 8/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337621 1.00 NOS3 (0.41) NOS3NOS2NOS1BACE1KLKB1
Hydrochloric Acid SCHEMBL17442571 0.98 NOS3 (0.41) NOS3NOS2NOS1BACE1KLKB1
Hydrochloric Acid SCHEMBL7823971 0.98 NOS3 (0.41) NOS3NOS2NOS1BACE1KLKB1
Trifluoroacetic Acid SCHEMBL18300447 0.83 KLKB1 (0.41) KLKB1
SCHEMBL7742237 0.83 HTR1D (0.47) NOS3NOS2NOS1BACE1
SCHEMBL14385061 0.83 NOS3 (0.39) NOS3NOS2NOS1BACE1
SCHEMBL9696219 0.83 NOS3 (0.45) NOS3NOS2NOS1BACE1KLKB1
Trifluoroacetic Acid SCHEMBL17221097 0.82 KLKB1 (0.40) KLKB1
SCHEMBL18301317 0.81 NOS3 (0.40) NOS3NOS2NOS1BACE1KLKB1
SCHEMBL18368343 0.80 POLB (0.38) NOS3NOS2NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396474-A Plasma kallikrein inhibitors 武田药品工业株式会社 2024-01-12 CN disclosed
CN-113004286-B Tricyclic compounds as plasma kallikrein inhibitors and uses thereof 成都康弘药业集团股份有限公司 2022-08-12 CN disclosed