SCHEMBL30001992

SCHEMBL30001992

CN1CCN(c2ccc(Nc3nc(-n4cnc5ccccc54)c4ccn(COCC[Si](C)(C)C)c4n3)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 6/20 0.60
MKNK1 Q9BUB5 2/20 0.52
PTK2 Q05397 2/20 0.47
EGFR P00533 2/20 0.43
LCK P06239 3/20 0.42
SRC P12931 3/20 0.42
BTK Q06187 2/20 0.41
ABL1 P00519 1/20 0.41
CDK4 P11802 3/20 0.40
AURKA O14965 2/20 0.40
KDM1A O60341 1/20 0.40
GLA P06280 1/20 0.40
ADRA2A P08913 1/20 0.40
SLC2A1 P11166 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CCND1 P24385 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30002763 0.78 MKNK1 (0.38) MKNK1
SCHEMBL28894262 0.78 MKNK1 (0.38) MKNK1
SCHEMBL15112625 0.76 FLT3 (0.41) PTK2EGFRBTKABL1CDK4
SCHEMBL30001563 0.75 TTK (1.00) TTKMKNK1PTK2
SCHEMBL15453521 0.75 EGFR (0.44) PTK2EGFRBTKCDK4AURKA
SCHEMBL23567042 0.74 JAK2 (0.53) PTK2EGFRJAK3
SCHEMBL15112637 0.73 BRD4 (0.44) PTK2EGFRCDK4CCND3JAK3
SCHEMBL15459980 0.72 EGFR (0.46) PTK2EGFRBTKCDK4AURKA
SCHEMBL15126299 0.71 JAK3 (0.53) EGFRSRCBTKADRA2ATYK2
SCHEMBL15453518 0.71 JAK3 (0.46) PTK2EGFRBTKCDK4AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115368364-B 7H-pyrrolo [2,3-d ] pyrimidine derivatives, preparation method and application thereof 四川大学 2024-07-16 CN disclosed
CN-115368364-A 7H-pyrrolo [2,3-d ] pyrimidine derivative and preparation method and application thereof 四川大学 2022-11-22 CN disclosed