SCHEMBL30003299

SCHEMBL30003299

CC(=O)Nc1c(C)c(F)cc(F)c1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.43
GAA P10253 4/20 0.43
KDM4E B2RXH2 2/20 0.43
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
ALDH1A1 P00352 4/20 0.39
HTT P42858 4/20 0.36
LMNA P02545 5/20 0.36
NPSR1 Q6W5P4 3/20 0.36
GALR2 O43603 1/20 0.36
MITF O75030 1/20 0.36
POLB P06746 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892238 1.00 MAPT (0.43) MAPTGAAKDM4EGRIN2DGRIN3B
SCHEMBL26981453 0.88 MAPT (0.43) MAPTGAAKDM4EGRIN2DGRIN3B
SCHEMBL21608252 0.83 MAPT (0.42) MAPTGAAKDM4EGRIN2DGRIN3B
SCHEMBL21684641 0.79 MAPT (0.44) MAPTGAAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL31569422 0.78 MAPT (0.43) MAPTGAAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL31569299 0.77 GAA (0.42) MAPTGAAKDM4EGRIN2DGRIN3B
SCHEMBL27795562 0.75 ALDH1A1 (0.47) MAPTGAAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL30002032 0.75 ALDH1A1 (0.47) MAPTGAAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL30946511 0.75 MAPT (0.40) MAPTGAAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL8112444 0.74 ALDH1A1 (0.40) MAPTGAAKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed