SCHEMBL30006036

SCHEMBL30006036

CN1C(=O)CCc2c(B3OC(C)(C)C(C)(C)O3)cccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.41
BTK Q06187 3/20 0.41
TRPV1 Q8NER1 8/20 0.34
HTR1A P08908 2/20 0.34
HTR1D P28221 2/20 0.34
HTR1B P28222 2/20 0.34
SLC6A4 P31645 2/20 0.34
KCNH2 Q12809 2/20 0.34
BRPF1 P55201 1/20 0.32
BRD4 O60885 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
CCKBR P32239 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
LPL P06858 1/20 0.30
LIPG Q9Y5X9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16110732 1.00 JAK2 (0.41) JAK2BTKTRPV1HTR1AHTR1D
SCHEMBL15332752 0.87 JAK2 (0.41) JAK2BTKBRPF1GABRA1GABRG2
SCHEMBL17713762 0.82 CYP11B1 (0.35) JAK2BTKTRPV1BRD4CYP11B1
SCHEMBL24428590 0.81 JAK2 (0.31) JAK2BTKBRD4
SCHEMBL17713696 0.81 JAK2 (0.35) JAK2BTKBRD4GABRG2GABRB3
SCHEMBL17546978 0.79 JAK2 (0.38) JAK2BTK
SCHEMBL19464228 0.78 JAK2 (0.38) JAK2BTKLPLLIPGP2RX7
SCHEMBL31707905 0.74 ALDH1A1 (0.37) JAK2BTKLPLLIPGP2RX7
SCHEMBL508291 0.74 ALDH1A1 (0.37) JAK2BTKLPLLIPGP2RX7
SCHEMBL1746088 0.73 NOTUM (0.43) JAK2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4090660-A1 QUINOXALINE DERIVATIVES Grünenthal GmbH (DE) 2022-11-23 EP disclosed