SCHEMBL30013596

SCHEMBL30013596

Nc1nc(N2CCOCC2)nc2c(-c3ccnnc3)cnn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
KDM4E B2RXH2 4/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PIK3CA P42336 10/20 0.42
MTOR P42345 7/20 0.42
PIK3R1 P27986 5/20 0.42
PIK3CG P48736 1/20 0.42
ERAP1 Q9NZ08 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CB P42338 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 2/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAP3K12 Q12852 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23497520 0.78 PIK3CA (0.43) NPC1RAB9APIK3CAMTORPIK3R1
SCHEMBL6894445 0.77 PIK3CA (0.50) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL30013171 0.74 PIK3CA (0.40) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL23497449 0.74 PIK3CA (0.46) RAB9AKDM4EMAPTPIK3CAMEN1
SCHEMBL23497499 0.74 ALDH1A1 (0.40) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL25140245 0.72 CSNK1E (0.51) KDM4EPIK3CDPIK3CBHPGD
SCHEMBL30013825 0.72 CSNK1E (0.51) KDM4EPIK3CDPIK3CBHPGD
SCHEMBL23508069 0.72 MTOR (0.50) PIK3CAMTORPIK3R1PIK3CGPIK3CD
SCHEMBL23497786 0.71 PIK3CA (0.45) KDM4EPIK3CAMTORPIK3R1ALDH1A1
SCHEMBL23508187 0.71 PIK3CA (0.38) KDM4EPIK3CAMTORPIK3R1PIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4073072-A1 PYRAZOLOTRIAZINES Bayer Aktiengesellschaft (DE) 2022-10-19 EP disclosed