SCHEMBL30019212

SCHEMBL30019212

CN1CCN(c2ccc(Nc3ncc4ccn(CC5CCOCC5)c4n3)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT6 P42226 6/20 0.62
CDK4 P11802 10/20 0.61
AURKA O14965 6/20 0.61
CDK1 P06493 2/20 0.61
INSR P06213 1/20 0.61
PDGFRB P09619 1/20 0.61
SRC P12931 1/20 0.61
PDGFRA P16234 1/20 0.61
FLT1 P17948 1/20 0.61
FLT4 P35916 1/20 0.61
KDR P35968 1/20 0.61
CDK7 P50613 1/20 0.61
NTRK2 Q16620 1/20 0.61
FGFR4 P22455 3/20 0.58
CCND1 P24385 4/20 0.56
CCND2 P30279 4/20 0.56
CCND3 P30281 4/20 0.56
CCNE2 O96020 2/20 0.55
CCNA2 P20248 2/20 0.55
CCNE1 P24864 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30019765 0.90 JAK2 (0.55) STAT6CDK4AURKACDK1INSR
SCHEMBL30017942 0.87 BTK (0.57) STAT6ABL1BTK
SCHEMBL30017946 0.86 TNK2 (0.63) STAT6CDK4AURKACDK1INSR
SCHEMBL30019218 0.86 TTK (0.61) CDK4INSRSRCCCND1
SCHEMBL30018989 0.84 CDK4 (0.56) CDK4AURKACDK1INSRPDGFRB
SCHEMBL30019432 0.83 TNK2 (0.57) STAT6SRC
SCHEMBL30017933 0.83 TNK2 (0.55) STAT6CDK4AURKACDK1INSR
SCHEMBL30019959 0.82 JAK1 (0.49) STAT6CDK4AURKA
SCHEMBL27844369 0.82 STAT6 (0.69) STAT6CDK4AURKACDK1INSR
SCHEMBL15163242 0.80 STAT6 (0.67) STAT6CDK4AURKACDK1INSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022226290-A1 2-PHENYLAMINO PYRROLOPYRIMIDINES AS ACK1 INHIBITORS H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2022-10-27 WO disclosed