SCHEMBL30020064

SCHEMBL30020064

CC(C)(C)OC(=O)N1CCC(CN2CCC(C(F)(F)F)CC2)CC1.FC(F)(F)C1CCN(CC2CCNCC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
RECQL P46063 1/20 0.38
EPHX1 P07099 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
GPR119 Q8TDV5 5/20 0.38
ACHE P22303 2/20 0.38
NR1H2 P55055 1/20 0.38
HTR4 Q13639 1/20 0.38
FAAH O00519 1/20 0.37
FPR2 P25090 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27347956 0.93 HPGD (0.45) KDM4EPKMHPGDRECQLEPHX1
SCHEMBL27307597 0.88 CACNA2D1 (0.45) KDM4EPKMHPGDRECQLACHE
SCHEMBL24480292 0.86 HPGD (0.46) KDM4EPKMHPGDRECQLEPHX1
SCHEMBL27144706 0.86 HPGD (0.57) KDM4EPKMHPGDRECQLEPHX1
SCHEMBL412749 0.85 HPGD (0.47) KDM4EPKMHPGDRECQLEPHX1
SCHEMBL2386299 0.85 CACNA2D1 (0.47) HPGDRECQLEPHX1MAPTNR1H2
Trifluoroacetic Acid SCHEMBL27848432 0.83 CACNA2D1 (0.45) KDM4EPKMHPGDMAPTGPR119
SCHEMBL27162825 0.82 KDM4E (0.42) KDM4EPKMHPGDRECQLEPHX1
SCHEMBL24480620 0.81 KDM4E (0.41) KDM4EPKMHPGDRECQLEPHX1
SCHEMBL27314016 0.81 KDM4E (0.41) KDM4EPKMHPGDGPR119FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4326724-A1 COMPOUND AS ADENOSINE A2A RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Chong Kun Dang Pharmaceutical Corp. (KR) 2024-02-28 EP disclosed
WO-2022224180-A1 COMPOUND AS ADENOSINE A2A RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITION COMPRISING SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2022-10-27 WO disclosed