SCHEMBL300214

SCHEMBL300214

CCCS(=O)(=O)c1ccc(-c2ccc(CC(C#N)NC(=O)C3CCOCC3)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.58
CTSK P43235 3/20 0.49
KCNH2 Q12809 1/20 0.45
LTB4R Q15722 1/20 0.45
LTB4R2 Q9NPC1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289950 0.81 CTSC (0.67) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL289987 0.81 CTSC (0.61) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL290568 0.81 CTSC (0.70) CTSCCTSK
SCHEMBL290339 0.81 CTSC (0.62) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL290045 0.79 CTSC (0.63) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL290172 0.78 CTSC (0.64) CTSCCTSK
SCHEMBL299918 0.76 CTSC (0.48) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL288812 0.75 CTSC (0.67) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL289448 0.74 CTSC (0.74) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL289447 0.74 CTSC (0.74) CTSCCTSKKCNH2LTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP claimed
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed