SCHEMBL30034874

SCHEMBL30034874

COc1ccc(-n2ccc3ccccc3c2=O)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.55
LMNA P02545 4/20 0.55
METAP2 P50579 1/20 0.52
G6PD P11413 1/20 0.50
HSD11B1 P28845 1/20 0.47
ALDH1A1 P00352 5/20 0.47
TP53 P04637 3/20 0.46
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
RAB9A P51151 3/20 0.45
KDM4E B2RXH2 2/20 0.45
NPC1 O15118 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
GRM1 Q13255 1/20 0.45
HPGD P15428 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28582077 1.00 MAPT (0.55) MAPTLMNAMETAP2G6PDHSD11B1
SCHEMBL28604399 0.85 KDM4E (0.56) ALDH1A1TP53KMT2AMEN1KDM4E
SCHEMBL2586137 0.84 ESRRA (0.47) MAPTLMNAMETAP2KMT2AMEN1
SCHEMBL4888172 0.84 KDM4E (0.47) ALDH1A1KDM4ERXFP1
SCHEMBL6185728 0.82 METAP2 (0.49) MAPTLMNAMETAP2G6PDALDH1A1
SCHEMBL29809422 0.82 METAP2 (0.49) MAPTLMNAMETAP2G6PDALDH1A1
SCHEMBL28593371 0.82 KDM4E (0.47) MAPTALDH1A1TP53KMT2AMEN1
SCHEMBL29431541 0.81 KDM4E (0.47) MAPTLMNAMETAP2G6PDALDH1A1
SCHEMBL2593323 0.81 KDM4E (0.47) MAPTLMNAMETAP2G6PDALDH1A1
SCHEMBL28565276 0.80 MAPT (0.41) MAPTLMNAMETAP2ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112876413-B Preparation and antiviral activity of 2- (isoquinoline-1 (2H) -ketone-4-yl) difluoro acetyl derivative 南开大学 2022-10-28 CN disclosed