SCHEMBL30046277

SCHEMBL30046277

CNc1cc(C)cc(F)c1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
MAPT P10636 6/20 0.42
LMNA P02545 4/20 0.42
NPC1 O15118 2/20 0.42
HTT P42858 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 2/20 0.42
MAPK1 P28482 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TLR9 Q9NR96 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
TSHR P16473 1/20 0.39
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27162953 1.00 ALDH1A1 (0.42) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL103325 0.84 MAPT (0.43) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL2274349 0.82 TSHR (0.50) ALDH1A1TSHRGRIN2DGRIN3BGRIN1
SCHEMBL16909268 0.81 MAPT (0.41) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL19980137 0.79 MAPT (0.43) ALDH1A1MAPTLMNANPC1RAB9A
SCHEMBL30045664 0.79 MAPT (0.42) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL30038957 0.79 ALDH1A1 (0.53) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL22154442 0.79 ALDH1A1 (0.53) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL27162629 0.79 MAPT (0.42) ALDH1A1MAPTLMNANPC1HTT
SCHEMBL27162701 0.78 MAPT (0.39) ALDH1A1MAPTLMNANPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4329749-A1 SMALL MOLECULE INHIBITORS OF KRAS G12C MUTANT Merck Sharp & Dohme LLC (US) 2024-03-06 EP disclosed
WO-2022232318-A1 SMALL MOLECULE INHIBITORS OF KRAS G12C MUTANT MERCK SHARP & DOHME CORP. (US) 2022-11-03 WO disclosed