SCHEMBL300486

SCHEMBL300486

O=C(N[C@H](CO)Cc1ccccc1)Oc1n[nH]c2c1CCCCC2Cc1cccc(Cl)c1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.65
EGFR P00533 2/20 0.40
PTGS2 P35354 1/20 0.35
PARP1 P09874 1/20 0.35
ADRB3 P13945 1/20 0.35
MME P08473 2/20 0.34
CTSV O60911 2/20 0.34
CTSL P07711 2/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 1/20 0.34
MMEL1 Q495T6 1/20 0.34
FFAR2 O15552 2/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300535 1.00 CNR2 (0.65) CNR2EGFRPTGS2PARP1ADRB3
SCHEMBL300497 0.90 CNR2 (0.78) CNR2
SCHEMBL300356 0.90 CNR2 (0.78) CNR2
SCHEMBL300479 0.90 CNR2 (0.78) CNR2
SCHEMBL300487 0.90 CNR2 (0.78) CNR2
SCHEMBL300533 0.90 CNR2 (0.78) CNR2
SCHEMBL300463 0.90 CNR2 (0.78) CNR2
SCHEMBL176480 0.88 CNR2 (0.80) CNR2EGFRPTGS2PARP1MME
SCHEMBL176535 0.88 CNR2 (0.80) CNR2EGFRPTGS2PARP1MME
SCHEMBL176651 0.79 CNR2 (1.00) CNR2CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed