SCHEMBL30069262

SCHEMBL30069262

C#CCOc1ccc(C=C(C(N)=O)c2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 1/20 0.49
MAPT P10636 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
GAA P10253 1/20 0.46
HDAC3 O15379 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
NCOR2 Q9Y618 2/20 0.46
MAOB P27338 3/20 0.43
AKR1C1 Q04828 1/20 0.43
LMNA P02545 2/20 0.43
MAOA P21397 2/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30480031 0.77 MAOB (0.39) KDM4EALDH1A1MAPTNPC1RAB9A
SCHEMBL23593943 0.76 AKR1C1 (0.70) KDM4EALDH1A1HPGDMAPTAKR1C1
SCHEMBL6689798 0.76 AKR1C1 (0.70) KDM4EALDH1A1HPGDMAPTAKR1C1
SCHEMBL2836206 0.76 AKR1C1 (0.70) KDM4EALDH1A1HPGDMAPTAKR1C1
SCHEMBL29006674 0.76 MAPT (0.68) ALDH1A1HPGDMAPTNPC1RAB9A
SCHEMBL29006676 0.76 MAPT (0.68) ALDH1A1HPGDMAPTNPC1RAB9A
SCHEMBL11529553 0.75 GAA (0.60) ALDH1A1MAPTRAB9AGAAMAOB
SCHEMBL11019288 0.72 AKR1C1 (0.55) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL11019290 0.72 AKR1C1 (0.55) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL20273256 0.72 PARP10 (0.59) ALDH1A1MAOBCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4351553-A1 NOVEL ANTI-FIBROTIC DRUGS Helmholtz Zentrum München Deutsches Forschungszentrum für Gesundheit und Umwelt GmbH (DE) 2024-04-17 EP disclosed
WO-2022258792-A1 NOVEL ANTI-FIBROTIC DRUGS Helmholtz Zentrum München - Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) (DE) 2022-12-15 WO disclosed