SCHEMBL30101633

SCHEMBL30101633

CCOC(=O)c1ccc2nc(N3CCC(NC(=O)c4ccc(Cl)c(Cl)c4)CC3)sc2c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 2/20 0.75
CCR3 P51677 1/20 0.58
SMN1; SMN2 Q16637 5/20 0.56
RAB9A P51151 5/20 0.56
NPC1 O15118 3/20 0.56
ALDH1A1 P00352 2/20 0.56
TMPRSS15 P98073 2/20 0.55
KDM4E B2RXH2 2/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
HPGD P15428 1/20 0.54
CYP2C19 P33261 1/20 0.54
MAPT P10636 4/20 0.53
POLB P06746 2/20 0.53
MITF O75030 1/20 0.51
TP53 P04637 1/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
KMT2A Q03164 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29123611 1.00 PCSK9 (0.75) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL30101767 0.89 PCSK9 (0.73) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL29123598 0.89 PCSK9 (0.73) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL30101747 0.87 PCSK9 (0.66) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL29123725 0.87 PCSK9 (0.66) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL30101699 0.87 PCSK9 (0.70) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL29123519 0.87 PCSK9 (0.70) PCSK9CCR3SMN1; SMN2RAB9ANPC1
SCHEMBL30101731 0.85 PCSK9 (1.00) PCSK9SMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL30101758 0.83 PCSK9 (0.76) PCSK9SMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL29123691 0.83 PCSK9 (0.76) PCSK9SMN1; SMN2RAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115109011-B Benzothiazole compound, preparation method and application 河北师范大学 2023-12-15 CN disclosed
CN-115109011-A Benzothiazole compound, preparation method and application 河北师范大学 2022-09-27 CN disclosed