SCHEMBL30101972

SCHEMBL30101972

O=c1[nH]c(-c2cccc(O)c2)nc2c(-c3cccnc3)nc(-c3ccc(C(F)(F)F)cc3)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 7/20 0.50
TNKS2 Q9H2K2 7/20 0.50
PARP1 P09874 4/20 0.50
PARP2 Q9UGN5 3/20 0.45
DGAT1 O75907 1/20 0.42
KCNH2 Q12809 1/20 0.42
WNT3A P56704 1/20 0.41
NPY5R Q15761 1/20 0.41
PIM1 P11309 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HPGD P15428 1/20 0.40
MAPT P10636 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KIT P10721 2/20 0.38
COMT P21964 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30101887 0.81 PIM1 (0.39) TNKSTNKS2PARP1PARP2DGAT1
SCHEMBL30101920 0.79 PIM1 (0.38) TNKSTNKS2PARP1PARP2DGAT1
SCHEMBL30101909 0.79 AHR (0.39) TNKSTNKS2PARP1PARP2DGAT1
SCHEMBL31472805 0.78 PIM1 (0.39) TNKSTNKS2PARP2DGAT1KCNH2
SCHEMBL30101858 0.78 AHR (0.38) TNKSTNKS2PARP1PARP2DGAT1
SCHEMBL30101960 0.78 PIM1 (0.37) TNKSTNKS2PARP1DGAT1KCNH2
SCHEMBL31472804 0.78 PIM1 (0.37) TNKSTNKS2PARP1PARP2DGAT1
SCHEMBL30101867 0.78 PIM1 (0.37) TNKSTNKS2PARP1DGAT1KCNH2
SCHEMBL23950529 0.78 PIM1 (0.45) PARP1DGAT1KCNH2NPY5RPIM1
SCHEMBL30101918 0.78 PIM1 (0.45) PARP1DGAT1KCNH2NPY5RPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN claimed
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN disclosed