SCHEMBL30102576

SCHEMBL30102576

COc1ccc(-c2cccc(-c3cc(OC)c(OC)c(OC)c3)n2)cc1Br

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.57
MAPT P10636 5/20 0.52
BRD4 O60885 1/20 0.49
KDM4E B2RXH2 4/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
NPC1 O15118 4/20 0.48
ALDH1A1 P00352 4/20 0.48
RAB9A P51151 3/20 0.48
HPGD P15428 2/20 0.48
RECQL P46063 1/20 0.48
GLA P06280 1/20 0.48
GAA P10253 1/20 0.48
ALOX12 P18054 1/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
TP53 P04637 1/20 0.47
THRB P10828 1/20 0.47
TUBB1 Q9H4B7 2/20 0.47
PDGFRB P09619 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28960772 1.00 HDAC8 (0.57) HDAC8MAPTBRD4KDM4ESMN1; SMN2
SCHEMBL18492964 0.88 HDAC8 (0.58) HDAC8MAPTBRD4KDM4ESMN1; SMN2
SCHEMBL17144470 0.86 HDAC8 (0.58) HDAC8MAPTBRD4KDM4ENPC1
SCHEMBL28960774 0.85 HDAC8 (0.60) HDAC8MAPTBRD4KDM4ENPC1
SCHEMBL28965201 0.84 HDAC8 (0.52) HDAC8MAPTBRD4KDM4ENPC1
SCHEMBL30102577 0.84 HDAC8 (0.52) HDAC8MAPTBRD4KDM4ENPC1
SCHEMBL30102580 0.82 HDAC8 (0.57) HDAC8MAPTKDM4ESMN1; SMN2NPC1
SCHEMBL17144926 0.82 HDAC8 (0.57) HDAC8MAPTKDM4ESMN1; SMN2NPC1
SCHEMBL16385293 0.82 MAPT (0.58) HDAC8MAPTKDM4ESMN1; SMN2NPC1
SCHEMBL17144925 0.81 BRD4 (0.54) HDAC8MAPTBRD4KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115572254-B 2, 6-Diaryl pyridine HDAC/Tubulin dual-function inhibitor and preparation method and application thereof 复旦大学 2025-04-01 CN disclosed
CN-115572254-A 2, 6-diaryl pyridine HDAC/Tubulin bifunctional inhibitor, preparation method and application 复旦大学 2023-01-06 CN disclosed