SCHEMBL30102580

SCHEMBL30102580

COc1ccc(-c2cccc(-c3cc(OC)c(OC)c(OC)c3)n2)cc1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.57
TUBB4A P04350 7/20 0.56
TUBB P07437 7/20 0.56
TUBA3C P0DPH7 7/20 0.56
TUBA1B P68363 7/20 0.56
TUBA4A P68366 7/20 0.56
TUBB4B P68371 7/20 0.56
TUBB3 Q13509 7/20 0.56
TUBB2A Q13885 7/20 0.56
TUBB8 Q3ZCM7 7/20 0.56
TUBA3E Q6PEY2 7/20 0.56
TUBA1A Q71U36 7/20 0.56
TUBA1C Q9BQE3 7/20 0.56
TUBB6 Q9BUF5 7/20 0.56
TUBB2B Q9BVA1 7/20 0.56
TUBB1 Q9H4B7 7/20 0.56
PDGFRB P09619 1/20 0.51
KIT P10721 1/20 0.51
KDR P35968 1/20 0.51
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17144926 1.00 HDAC8 (0.57) HDAC8TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL18492964 0.88 HDAC8 (0.58) HDAC8TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL17144470 0.86 HDAC8 (0.58) HDAC8PDGFRBKITKDRKDM4E
SCHEMBL17144844 0.85 PDGFRB (0.60) HDAC8PDGFRBKITKDRALDH1A1
SCHEMBL30102576 0.82 HDAC8 (0.57) HDAC8TUBB1PDGFRBKITKDR
SCHEMBL28960772 0.82 HDAC8 (0.57) HDAC8TUBB1PDGFRBKITKDR
SCHEMBL17144923 0.80 PDGFRB (0.59) HDAC8TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL17144996 0.79 KDM4E (0.65) KDM4EMEN1NPC1ALDH1A1TP53
SCHEMBL28960774 0.79 HDAC8 (0.60) HDAC8TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL30102579 0.78 CYP1A1 (0.50) HDAC8KDM4EMEN1NPC1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115572254-A 2, 6-diaryl pyridine HDAC/Tubulin bifunctional inhibitor, preparation method and application 复旦大学 2023-01-06 CN disclosed