SCHEMBL30104848

SCHEMBL30104848

O=C1NCCn2c1cc1cc(C(F)(F)F)ccc12

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.49
CYP2D6 P10635 1/20 0.48
RPS6KA2 Q15349 2/20 0.46
PARP1 P09874 5/20 0.44
PARP10 Q53GL7 1/20 0.43
RPS6KA3 P51812 2/20 0.41
MAPKAPK2 P49137 2/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29153647 1.00 HRH3 (0.49) HRH3CYP2D6RPS6KA2PARP1PARP10
SCHEMBL19187485 0.81 HRH3 (0.52) HRH3CYP2D6RPS6KA2PARP1PARP10
SCHEMBL2980522 0.78 HRH3 (0.52) HRH3CYP2D6RPS6KA2PARP1RPS6KA3
SCHEMBL38652638 0.78 HRH3 (0.52) HRH3CYP2D6RPS6KA2PARP1PARP10
SCHEMBL38652559 0.78 HRH3 (0.52) HRH3CYP2D6RPS6KA2PARP1RPS6KA3
SCHEMBL2160684 0.78 HRH3 (0.54) HRH3CYP2D6RPS6KA2PARP1RPS6KA3
SCHEMBL1393632 0.76 RPS6KA3 (0.53) HRH3CYP2D6RPS6KA2PARP1RPS6KA3
SCHEMBL30172384 0.76 RPS6KA3 (0.53) HRH3CYP2D6RPS6KA2PARP1RPS6KA3
SCHEMBL24640536 0.76 CDK4 (0.42) HRH3CYP2D6RPS6KA2PARP1RPS6KA3
SCHEMBL30104808 0.76 RPS6KA2 (0.42) HRH3CYP2D6RPS6KA2PARP1RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396485-A PARP7 inhibitors 轩竹生物科技股份有限公司 2024-01-12 CN disclosed
WO-2022247839-A1 PARP7 INHIBITOR 山东轩竹医药科技有限公司 2022-12-01 WO disclosed