SCHEMBL30108028

SCHEMBL30108028

Nc1nc(-c2ccco2)cc(-n2nnc3cc(Oc4ccccc4)ccc32)n1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ADORA2A P29274 6/20 0.38
ADORA2B P29275 4/20 0.38
ADORA1 P30542 4/20 0.38
TNK2 Q07912 1/20 0.37
ADORA3 P0DMS8 3/20 0.37
PTGS1 P23219 2/20 0.37
NPC1 O15118 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGS2 P35354 1/20 0.35
MCL1 Q07820 2/20 0.35
SMARCA2 P51531 1/20 0.35
PBRM1 Q86U86 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30107951 0.88 PTGS1 (0.46) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30107991 0.88 HSD17B10 (0.38) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30107986 0.88 HSD17B10 (0.38) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30107980 0.87 ROCK1 (0.45) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30107943 0.86 KDM4E (0.37) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30108012 0.84 TSHR (0.58) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30108046 0.83 KDM4E (0.39) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30107959 0.82 KDM4E (0.44) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30108023 0.81 PTGS1 (0.47) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL30108014 0.80 KDM4E (0.42) KDM4EALDH1A1GAAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed