SCHEMBL30107951

SCHEMBL30107951

COc1ccc2c(c1)nnn2-c1cc(-c2ccco2)nc(N)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46
THRB P10828 1/20 0.46
ALOX12 P18054 1/20 0.46
PTPN7 P35236 1/20 0.46
HTT P42858 1/20 0.46
RECQL P46063 1/20 0.46
RAB9A P51151 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
MCL1 Q07820 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ADORA2A P29274 5/20 0.45
ADORA1 P30542 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108028 0.88 KDM4E (0.43) PTGS1PTGS2KDM4EALDH1A1HPGD
SCHEMBL30107973 0.88 KDM4E (0.46) PTGS1PTGS2KDM4EALDH1A1HPGD
SCHEMBL30107980 0.84 ROCK1 (0.45) PTGS1PTGS2KDM4EALDH1A1HPGD
SCHEMBL30108046 0.84 KDM4E (0.39) PTGS1PTGS2KDM4EALDH1A1HPGD
SCHEMBL30107959 0.84 KDM4E (0.44) KDM4EALDH1A1HPGDADORA2AADORA1
SCHEMBL30107986 0.84 HSD17B10 (0.38) PTGS1PTGS2KDM4EALDH1A1HPGD
SCHEMBL30107991 0.84 HSD17B10 (0.38) PTGS1PTGS2KDM4EALDH1A1HPGD
SCHEMBL30108012 0.83 TSHR (0.58) PTGS1KDM4EALDH1A1HPGDPOLB
SCHEMBL30107994 0.83 PTGS1 (0.50) PTGS1KDM4EALDH1A1HPGDMEN1
SCHEMBL30108014 0.81 KDM4E (0.42) KDM4EALDH1A1HPGDADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed