SCHEMBL30108079

SCHEMBL30108079

CSc1nc(N)c(Br)c(Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
HSP90AB1 P08238 2/20 0.39
ABCB1 P08183 2/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSP90AA1 P07900 3/20 0.35
LMNA P02545 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15904101 1.00 KMT2A (0.41) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9
SCHEMBL22055448 0.84 HSP90AB1 (0.46) KMT2AHSP90AB1ABCB1HSP90AA1LMNA
SCHEMBL11191903 0.80 HSP90AB1 (0.40) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9
SCHEMBL11225658 0.80 HSP90AB1 (0.40) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9
SCHEMBL29439810 0.78 CYP1A2 (0.39) KMT2AHSP90AB1CYP1A2CYP2C9CYP2C19
SCHEMBL22715908 0.78 CYP1A2 (0.39) KMT2AHSP90AB1CYP1A2CYP2C9CYP2C19
SCHEMBL6034037 0.78 ABCB1 (0.46) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL11429110 0.77 ABCB1 (0.44) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9
SCHEMBL18893671 0.77 HSP90AB1 (0.38) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9
SCHEMBL719751 0.77 HSP90AB1 (0.38) KMT2AHSP90AB1ABCB1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683033-B Substituted alkynyl heterocyclic compounds Capital Pharmaceutical Holdings (Beijing) Co.,Ltd. (CN) 2026-05-26 CN disclosed
CN-113880842-B Substituted alkynyl heterocyclic compounds 首药控股(北京)股份有限公司 2025-02-25 CN disclosed
CN-113004282-B Substituted alkynyl heterocyclic compounds 首药控股(北京)股份有限公司 2024-05-24 CN disclosed
CN-117683033-A Substituted alkynyl heterocyclic compounds 首药控股(北京)股份有限公司 2024-03-12 CN disclosed
CN-110290808-B 1- (4-amino-5-bromo-6- (1H-pyrazol-1-yl) pyrimidin-2-yl) -1H-pyrazol-4-ol and use thereof in the treatment of cancer 诺华股份有限公司 2023-07-11 CN disclosed
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed