SCHEMBL29439810

SCHEMBL29439810

CSc1nc(C)c(Br)c(Cl)n1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
PKM P14618 1/20 0.35
HSP90AB1 P08238 1/20 0.34
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
LMNA P02545 1/20 0.32
NR1I2 O75469 1/20 0.31
AHR P35869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22715908 1.00 CYP1A2 (0.39) CYP1A2CYP2C9CYP2C19KMT2APKM
SCHEMBL30108079 0.78 KMT2A (0.41) CYP1A2CYP2C9CYP2C19KMT2AHSP90AB1
SCHEMBL15904101 0.78 KMT2A (0.41) CYP1A2CYP2C9CYP2C19KMT2AHSP90AB1
SCHEMBL12712135 0.77 KMT2A (0.38) CYP1A2CYP2C9CYP2C19KMT2APKM
SCHEMBL11166832 0.77 LMNA (0.39) CYP1A2CYP2C9CYP2C19KMT2APKM
SCHEMBL1935371 0.74 KMT2A (0.36) CYP1A2CYP2C9CYP2C19KMT2APKM
SCHEMBL75623 0.74 PDE10A (0.41) CYP1A2CYP2C9CYP2C19KMT2APKM
SCHEMBL31718366 0.72 LMNA (0.37) LMNANR1I2AHR
SCHEMBL29350081 0.72 LMNA (0.37) ALDH1A1LMNANR1I2AHR
SCHEMBL4068928 0.72 LMNA (0.37) ALDH1A1LMNANR1I2AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed