SCHEMBL30108147

SCHEMBL30108147

COc1cc(F)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(Nc2ccc(CC(N)=O)cc2OC)n1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 11/20 0.55
LRRK2 Q5S007 4/20 0.50
MAPK3 P27361 2/20 0.49
ZAP70 P43403 2/20 0.48
INSR P06213 4/20 0.47
IGF1R P08069 1/20 0.47
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
MAPK10 P53779 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108145 0.95 ALK (0.61) ALKLRRK2MAPK3INSRIGF1R
SCHEMBL30108134 0.88 ALK (0.52) ALKINSRIGF1RMAPK8MAPK9
SCHEMBL30108139 0.88 ALK (0.51) ALKINSRIGF1RMAPK8MAPK9
SCHEMBL28728655 0.87 LRRK2 (0.51) ALKLRRK2MAPK3ZAP70INSR
SCHEMBL30108143 0.86 ALK (0.57) ALKINSRIGF1RMAPK8MAPK9
SCHEMBL28728617 0.84 ALK (0.59) ALKMAPK3ZAP70INSR
SCHEMBL28728854 0.84 LRRK2 (0.47) ALKLRRK2MAPK3ZAP70INSR
SCHEMBL29594720 0.82 ALK (0.49) ALKLRRK2MAPK3ZAP70INSR
SCHEMBL25449374 0.80 ZAP70 (0.47) ALKLRRK2MAPK3ZAP70INSR
SCHEMBL28728761 0.80 ALK (0.60) ALKMAPK3INSRIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394974-B Polysubstituted triaryl macrocyclic compounds and uses thereof 中国药科大学 2022-12-06 CN disclosed