SCHEMBL30108145

SCHEMBL30108145

COc1cc(F)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(Nc2cc(CC(N)=O)ccc2OC)n1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 18/20 0.61
INSR P06213 8/20 0.52
LRRK2 Q5S007 1/20 0.46
IGF1R P08069 1/20 0.46
MAPK3 P27361 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108147 0.95 ALK (0.55) ALKINSRLRRK2IGF1RMAPK3
SCHEMBL30108134 0.93 ALK (0.52) ALKINSRIGF1R
SCHEMBL30108139 0.93 ALK (0.51) ALKINSRIGF1R
SCHEMBL30108143 0.91 ALK (0.57) ALKINSRIGF1R
SCHEMBL28728854 0.87 LRRK2 (0.47) ALKINSRLRRK2IGF1RMAPK3
SCHEMBL29594720 0.86 ALK (0.49) ALKINSRLRRK2IGF1RMAPK3
SCHEMBL30108135 0.85 ALK (0.53) ALKINSRLRRK2IGF1R
SCHEMBL30108148 0.84 ALK (0.42) ALKINSRLRRK2IGF1R
SCHEMBL29595331 0.84 ALK (0.60) ALKINSRIGF1RMAPK3
SCHEMBL28728655 0.84 LRRK2 (0.51) ALKINSRLRRK2IGF1RMAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394974-B Polysubstituted triaryl macrocyclic compounds and uses thereof 中国药科大学 2022-12-06 CN disclosed