SCHEMBL30111348

SCHEMBL30111348

COc1cccc(-c2cc(N)c3ccccc3n2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.67
ADORA2A P29274 1/20 0.63
TOP1 P11387 1/20 0.59
ABCB1 P08183 1/20 0.57
ABCG2 Q9UNQ0 1/20 0.57
CYP1A2 P05177 3/20 0.57
CYP3A4 P08684 3/20 0.57
CYP2C9 P11712 3/20 0.57
CYP2B6 P20813 2/20 0.57
AHR P35869 2/20 0.57
NR1I3 Q14994 2/20 0.57
VDR P11473 1/20 0.57
ACACA Q13085 1/20 0.56
KMT2A Q03164 6/20 0.54
HPGD P15428 6/20 0.54
SMN1; SMN2 Q16637 5/20 0.54
MEN1 O00255 4/20 0.54
LMNA P02545 4/20 0.54
TP53 P04637 1/20 0.54
ALDH1A1 P00352 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4914795 0.89 KDM4E (0.59) ACHEADORA2ATOP1ABCB1ABCG2
SCHEMBL28510601 0.87 ACHE (0.69) ACHEADORA2ATOP1ABCB1ABCG2
SCHEMBL4817642 0.86 KDM4E (0.65) ACHEADORA2ATOP1ABCB1ABCG2
SCHEMBL28506567 0.85 KDM4E (0.71) ACHEADORA2ACYP1A2ACACAHPGD
Hydrochloric Acid SCHEMBL29874770 0.84 KDM4E (0.69) ACHEADORA2ACYP1A2ACACAHPGD
Hydrochloric Acid SCHEMBL29874996 0.84 KDM4E (0.69) ACHEADORA2ACYP1A2ACACAHPGD
Hydrochloric Acid SCHEMBL29874842 0.84 KDM4E (0.69) ACHEADORA2ACYP1A2ACACAHPGD
SCHEMBL4252226 0.84 TOP1 (0.51) ACHEADORA2ATOP1ABCB1ABCG2
SCHEMBL4246554 0.84 KDM4E (0.51) ACHEADORA2ATOP1CYP1A2CYP3A4
Ammonia Solution, Strong SCHEMBL4825130 0.84 MAPT (0.51) ACHEADORA2ATOP1ABCB1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4096666-A1 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE, NEURODEVELOPMENTAL, MYODEGENERATIVE, AND LYSOSOMAL STORAGE DISORDERS Georgetown University (US) 2022-12-07 EP disclosed