SCHEMBL30120738

SCHEMBL30120738

CN(C(=O)CCl)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.41
HTT P42858 4/20 0.41
RAB9A P51151 3/20 0.41
APEX1 P27695 1/20 0.41
LMNA P02545 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KMT2A Q03164 2/20 0.39
AGPAT2 O15120 1/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
OPRK1 P41145 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23723627 1.00 ALDH1A1 (0.48) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL15378617 0.86 AGPAT2 (0.50) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL11399589 0.86 ALDH1A1 (0.48) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL26660394 0.85 ALDH1A1 (0.55) ALDH1A1HTTRAB9ASMN1; SMN2KMT2A
SCHEMBL17336369 0.84 ALDH1A1 (0.47) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL19341421 0.83 ALDH1A1 (0.56) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL9823820 0.83 ALDH1A1 (0.52) ALDH1A1HDAC3HDAC1HDAC2HDAC6
SCHEMBL19879909 0.82 ALDH1A1 (0.48) ALDH1A1HTTRAB9ALMNASMN1; SMN2
SCHEMBL17336404 0.82 ALDH1A1 (0.43) ALDH1A1HDAC6HTTSMN1; SMN2
SCHEMBL23723732 0.81 ALDH1A1 (0.48) ALDH1A1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4100015-A1 COMBINATION THERAPY FOR TREATING MPS1 Gain Therapeutics SA (CH) 2022-12-14 EP disclosed
CN-115397423-A Combination therapy for the treatment of MPS1 增益治疗股份有限公司 2022-11-25 CN disclosed