SCHEMBL30123501

SCHEMBL30123501

Cc1cccc(C#Cc2ccc(-c3c(-c4ccncc4)cnn3C)cc2)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.59
PDE10A Q9Y233 9/20 0.56
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
CYP2C19 P33261 1/20 0.48
THPO P40225 1/20 0.48
KMT2A Q03164 1/20 0.48
GRIN2B Q13224 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15733793 1.00 GRM5 (0.59) GRM5PDE10ANPC1RAB9ASMN1; SMN2
SCHEMBL15022079 0.83 PDE10A (0.51) PDE10APDE4BPDE3BPDE3A
SCHEMBL15735320 0.82 GRM5 (0.51) GRM5PDE10ANPC1RAB9ASMN1; SMN2
SCHEMBL15745980 0.80 BRAF (0.47) PDE10APDE4BPDE3BPDE3A
SCHEMBL30123641 0.78 PDE10A (0.78) GRM5PDE10ANPC1RAB9ASMN1; SMN2
SCHEMBL15043339 0.78 PDE10A (0.78) GRM5PDE10ANPC1RAB9ASMN1; SMN2
SCHEMBL15733106 0.75 PDE10A (0.71) GRM5PDE10ANPC1RAB9ASMN1; SMN2
SCHEMBL15735281 0.72 PDE10A (1.00) GRM5PDE10ANPC1RAB9ASMN1; SMN2
SCHEMBL4724002 0.70 BRAF (0.53) PDE10APDE4BPDE3BPDE3A
SCHEMBL8119242 0.69 PRMT5 (0.48) PDE10ANPC1RAB9AKMT2APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115484938-A Composition and use thereof 博善人工智能剑桥有限公司 2022-12-16 CN disclosed