SCHEMBL30123641

SCHEMBL30123641

Cc1cccc(C#Cc2ccc(-c3nn(C)cc3-c3ccncc3)cc2)n1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 10/20 0.78
GRM5 P41594 3/20 0.58
MAPK14 Q16539 2/20 0.53
MAPK13 O15264 1/20 0.53
CSNK1D P48730 1/20 0.53
CSNK1E P49674 1/20 0.53
MAPK12 P53778 1/20 0.53
MAPK11 Q15759 1/20 0.53
BRAF P15056 5/20 0.49
MAPK3 P27361 1/20 0.48
MAPK1 P28482 1/20 0.48
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15043339 1.00 PDE10A (0.78) PDE10AGRM5MAPK14MAPK13CSNK1D
SCHEMBL30123690 0.89 PDE10A (0.77) PDE10AGRM5MAPK14MAPK13CSNK1D
SCHEMBL15733668 0.89 PDE10A (0.77) PDE10AGRM5MAPK14MAPK13CSNK1D
SCHEMBL15735701 0.88 PDE10A (1.00) PDE10AGRM5MAPK14BRAFKDM4E
SCHEMBL15734464 0.88 PDE10A (0.77) PDE10AGRM5MAPK14MAPK13CSNK1D
SCHEMBL30122884 0.88 PDE10A (1.00) PDE10AGRM5MAPK14BRAFKDM4E
SCHEMBL15734407 0.88 PDE10A (1.00) PDE10AGRM5MAPK14KDM4EMEN1
SCHEMBL30122927 0.87 PDE10A (1.00) PDE10AGRM5MAPK14KDM4EMEN1
SCHEMBL15734191 0.87 PDE10A (1.00) PDE10AGRM5MAPK14KDM4EMEN1
SCHEMBL15022282 0.86 PDE10A (0.59) PDE10AMAPK14MAPK13CSNK1DCSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115484938-A Composition and use thereof 博善人工智能剑桥有限公司 2022-12-16 CN disclosed