SCHEMBL30125317

SCHEMBL30125317

CC(C)C(CNc1nc(-n2cccc2)nc2ccccc12)N1CCN(C)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 6/20 0.54
PDE5A O76074 5/20 0.54
HTR3A P46098 2/20 0.47
SLC6A3 Q01959 2/20 0.46
KDM4E B2RXH2 4/20 0.42
KMT2A Q03164 2/20 0.42
HSD17B10 Q99714 2/20 0.42
GAA P10253 2/20 0.42
PTGS1 P23219 1/20 0.42
TBXAS1 P24557 1/20 0.42
PTGS2 P35354 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
MEN1 O00255 1/20 0.42
GLA P06280 1/20 0.42
TSHR P16473 1/20 0.42
NPY1R P25929 1/20 0.42
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23723290 1.00 HRH4 (0.54) HRH4PDE5AHTR3ASLC6A3KDM4E
SCHEMBL23747916 0.87 HRH4 (0.59) HRH4PDE5AHTR3AKDM4EKMT2A
SCHEMBL23723346 0.84 PDE5A (0.48) HRH4PDE5AHTR3ASLC6A3KDM4E
SCHEMBL30125141 0.84 PDE5A (0.48) HRH4PDE5AHTR3ASLC6A3KDM4E
SCHEMBL23747915 0.79 CYP1A2 (0.57) SLC6A3KDM4EKMT2AHSD17B10MAPT
SCHEMBL23747961 0.79 HRH4 (0.63) HRH4PDE5AHTR3AKDM4EHSD17B10
SCHEMBL23747842 0.78 GBA1 (0.55) PDE5ASLC6A3KDM4EKMT2AMAPT
SCHEMBL23747909 0.78 PDE5A (0.54) HRH4PDE5ASLC6A3KMT2AMAPT
SCHEMBL23747914 0.78 SLC6A3 (0.54) HRH4PDE5ASLC6A3HSD17B10ALOX15
SCHEMBL23723287 0.78 SLC6A3 (0.54) HRH4PDE5ASLC6A3ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4100395-A1 QUINAZOLINE COMPOUNDS AND THE USE THEREOF IN THE TREATMENT OF CANCER Trobio Therapeutics Pty Ltd (AU) 2022-12-14 EP disclosed