SCHEMBL30131372

SCHEMBL30131372

C#CCNC(=O)c1ncccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
EGLN2 Q96KS0 1/20 0.44
FTO Q9C0B1 1/20 0.44
RIPK1 Q13546 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GRM1 Q13255 1/20 0.40
GAA P10253 1/20 0.40
MAPK8 P45983 1/20 0.39
CTSA P10619 1/20 0.39
GPX4 P36969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30131385 0.86 EGLN1 (0.52) ALDH1A1EGLN2FTONPC1RAB9A
SCHEMBL15711407 0.84 RIPK1 (0.46) EGLN2FTORIPK1KMT2ACA12
SCHEMBL30131408 0.84 NPC1 (0.47) ALDH1A1EGLN2FTORIPK1NPC1
SCHEMBL30131325 0.81 PDE4B (0.48) EGLN2FTORIPK1NPC1RAB9A
SCHEMBL9210564 0.81 KDM4E (0.46) ALDH1A1EGLN2FTORIPK1NPC1
SCHEMBL11788023 0.80 SMN1; SMN2 (0.56) ALDH1A1NPC1POLBHPGDMEN1
SCHEMBL30131499 0.80 EGLN2 (0.43) ALDH1A1EGLN2FTONPC1RAB9A
SCHEMBL29459608 0.79 POLB (0.47) EGLN2FTONPC1RAB9APOLB
SCHEMBL30131667 0.79 HPGD (0.56) ALDH1A1NPC1RAB9AHPGDMEN1
SCHEMBL30131475 0.79 HPGD (0.60) ALDH1A1NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117715898-A Six-membered aryl or heteroaryl amide compound, composition and application thereof 贝达药业股份有限公司 2024-03-15 CN claimed
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO claimed
CN-117715898-A Six-membered aryl or heteroaryl amide compound, composition and application thereof 贝达药业股份有限公司 2024-03-15 CN disclosed
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO disclosed