SCHEMBL30132099

SCHEMBL30132099

COc1ccccc1-n1ncc2c(O)nc(CN(C)CC(=O)N(C)c3ccccc3Cl)nc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 5/20 0.38
ALDH1A1 P00352 3/20 0.38
POLB P06746 1/20 0.38
USP2 O75604 1/20 0.35
GLA P06280 1/20 0.35
SCN5A Q14524 2/20 0.34
SCN9A Q15858 2/20 0.34
SLC2A1 P11166 1/20 0.34
SLC2A2 P11168 1/20 0.34
SLC2A3 P11169 1/20 0.34
RAB9A P51151 2/20 0.34
TSHR P16473 2/20 0.34
S1PR2 O95136 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPK14 Q16539 1/20 0.34
PDE5A O76074 3/20 0.33
PDE1B Q01064 3/20 0.33
PDE4D Q08499 3/20 0.33
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23723650 1.00 PDE9A (0.38) PDE9AALDH1A1POLBUSP2GLA
SCHEMBL23723619 0.89 GRM5 (0.41) PDE9AALDH1A1POLBTSHRSMN1; SMN2
SCHEMBL30132061 0.89 GRM5 (0.41) PDE9AALDH1A1POLBTSHRSMN1; SMN2
SCHEMBL30132094 0.87 TSHR (0.42) PDE9AALDH1A1POLBRAB9ATSHR
SCHEMBL23723520 0.87 TSHR (0.42) PDE9AALDH1A1POLBRAB9ATSHR
SCHEMBL23723808 0.86 GRM1 (0.38) ALDH1A1RAB9ATSHRSMN1; SMN2NPC1
SCHEMBL30132062 0.86 GRM1 (0.38) ALDH1A1RAB9ATSHRSMN1; SMN2NPC1
SCHEMBL23723609 0.85 SMN1; SMN2 (0.42) PDE9AALDH1A1POLBTSHRSMN1; SMN2
SCHEMBL30132074 0.85 SMN1; SMN2 (0.42) PDE9AALDH1A1POLBTSHRSMN1; SMN2
SCHEMBL23723692 0.84 MAPT (0.40) ALDH1A1POLBRAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4100015-A1 COMBINATION THERAPY FOR TREATING MPS1 Gain Therapeutics SA (CH) 2022-12-14 EP disclosed