SCHEMBL30132100

SCHEMBL30132100

Cc1ccc2nc(CN(C)CC(=O)N3CCc4ccccc43)[nH]c(=O)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.54
MAPT P10636 5/20 0.52
LMNA P02545 3/20 0.47
TSHR P16473 2/20 0.47
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NPC1 O15118 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HTT P42858 2/20 0.46
KDM4E B2RXH2 2/20 0.46
GBA1 P04062 1/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 3/20 0.44
ALPL P05186 1/20 0.44
ALPI P09923 1/20 0.44
KMT2A Q03164 1/20 0.44
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
GLA P06280 1/20 0.43
CDK4 P11802 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26521632 1.00 PARP1 (0.54) PARP1MAPTLMNATSHRRAB9A
SCHEMBL26521647 0.93 PARP1 (0.54) PARP1MAPTLMNATSHRRAB9A
SCHEMBL23723559 0.90 ALDH1A1 (0.52) PARP1MAPTLMNATSHRRAB9A
SCHEMBL26524354 0.85 MAPT (0.51) PARP1MAPTLMNATSHRALDH1A1
SCHEMBL23723748 0.85 MAPT (0.51) PARP1MAPTLMNATSHRRAB9A
SCHEMBL23749976 0.84 PARP1 (0.61) PARP1MAPTLMNATSHRSMN1; SMN2
SCHEMBL26521585 0.83 TSHR (0.48) PARP1MAPTLMNATSHRRAB9A
SCHEMBL30132126 0.83 TSHR (0.48) PARP1MAPTLMNATSHRRAB9A
SCHEMBL26521975 0.80 MAPT (0.46) MAPTTSHRRAB9ASMN1; SMN2NPC1
SCHEMBL23882083 0.78 ALDH1A1 (0.51) PARP1MAPTLMNARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4100015-A1 COMBINATION THERAPY FOR TREATING MPS1 Gain Therapeutics SA (CH) 2022-12-14 EP disclosed